2. GPCR/G Protein Neuronal Signaling
  3. MCHR1 (GPR24)
  4. MCHR1 antagonist 1

MCHR1 antagonist 1 是一种选择性的黑色素浓集激素 1 型受体 (melanin concentrating hormone-1 receptor) 拮抗剂，对人 MCH1 受体的 Kb 和 Ki 值分别为 1 nM 和 4 nM，在降低体重方面可能起作用。

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MCHR1 antagonist 1 Chemical Structure

MCHR1 antagonist 1 Chemical Structure

CAS No. : 391610-37-0

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MCHR1 antagonist 1 相关抗体

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  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

MCHR1 antagonist 1 is a selective antagonist of melanin concentrating hormone-1 (MCH1) receptor, with a Kb of 1 nM and a Ki of 4 nM at human MCH1, and may be used to reduce the body mass.

IC50 & Target

Kb: 1 nM (Human MCH1)[1]
Ki: 4 nM (Human MCH1)[1]
体外研究
(In Vitro)

MCHR1 antagonist 1 shows potent activities against melanin concentrating hormone-1 receptor, but less potent against human MCH1, NPY1, NPY5, GALR1, GALR2, GALR3, and rat 5HT2C receptors, with Kis of >50000 nM[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

MCHR1 antagonist 1 相关抗体:
分子量

557.59

Formula

C28H33F2N5O5
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

MCHR1 antagonist 1 相关分类

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

MCHR1 antagonist 1391610-37-0MCHR1 (GPR24)Melanin concentrating hormone receptor 1Inhibitorinhibitorinhibit

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